HU-210 is a synthetic agonist analog of .DELTA.9-THC, which is the primary psychoactive component of marijuana. HU-210 is a potent central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptor agonist. It binds to neuroblastoma cell membrane CB1 receptors with about the same affinity as CP 55,940. In mouse behavior models (hypothermia, analgesia, hypoactivity, and catalepsy) the ED50 is 5-20 ug/kg.
产品描述
A synthetic agonist analog of Δ9-THC, which is the primary psychoactive component of marijuana; a potent CB1 and CB2 receptor agonist that binds to neuroblastoma cell membrane CB1 receptors with about the same affinity as CP 55,940; demonstrates ED50 values of 5-20 ug/kg in murine hypothermia, analgesia, hypoactivity, and catalepsy models